771
Unique InChIKey
1402
Unique Sequence
6157
EC50 Parameter
45
Unique DOI
Results
Showing 38581 to 38610 of 77611 results
| mus musculus | Olfr43 | Q7TRX1 | A108G_V205I | MREENESSTTDFTLL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S9 | |
| mus musculus | Olfr43 | Q7TRX1 | A152G_V205I | MREENESSTTDFTLL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S9 | |
| mus musculus | Olfr43 | Q7TRX1 | A108G_A152G_V205I | MREENESSTTDFTLL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S9 | |
| mus musculus | Olfr2 | Q9QWU6 | MERRNHTGRVSEFVL ... | Decanal | 8175 | KSMVZQYAVGTKIV-UHFFFAOYSA-N | CCCCCCCCCC=O | mono | 1 | norm_rec | 30 | uM | 28 | Ca2+ | OSN | liquid | ex vivo | olf | A pharmacological profile of t ... | https://doi.org/10.1113/jphysi ... | Table_1 | |||||||
| mus musculus | Olfr43 | Q7TRX1 | G106A_A108G_A152G_V205I | MREENESSTTDFTLL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 1 | ec50 | 235.6 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S9 | |
| bos taurus | OR1A1C | E1BBG9 | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | ||
| bos taurus | OR1A1C | E1BBG9 | L105I | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | |
| bos taurus | OR1A1C | E1BBG9 | V205I | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 1 | ec50 | >300 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | |
| bos taurus | OR1A1C | E1BBG9 | I277T | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 1 | ec50 | 581.15 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | |
| bos taurus | OR1A1C | E1BBG9 | L105I_V205I | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 1 | ec50 | >400 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | |
| bos taurus | OR1A1C | E1BBG9 | L105I_I277T | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | |
| bos taurus | OR1A1C | E1BBG9 | V205I_I277T | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 1 | ec50 | 584.19 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | |
| bos taurus | OR1A1C | E1BBG9 | L105I_V205I_I277T | MREDNQSSTLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 1 | ec50 | >1000 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Table_S10 | |
| pan troglodytes | OR1A1 | Q9TUA7 | MRENNQSSTLEFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 1 | ec50 | >100 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_2D | ||
| pan troglodytes | OR1A1 | Q9TUA7 | MRENNQSSTLEFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 1 | ec50 | >100 | uM | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_2D | ||
| homo sapiens | OR1A2 | Q9Y585 | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_2C | ||
| homo sapiens | OR1A2 | Q9Y585 | MKKENQSFNLDFILL ... | (S)-(+)-Carvone | 16724 | ULDHMXUKGWMISQ-VIFPVBQESA-N | CC1=CC[C@@H](CC1=O)C(=C)C | mono | 0 | ec50 | n.d | n.d | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_2C | ||
| homo sapiens | OR1A2 | Q9Y585 | A108G | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | K109N | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | V205I | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | T254V | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | V277T | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_K109N | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_V205I | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_K109N_V205I | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_K109N_T254V | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_K109N_V205I_T254V | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_K109N_V205I_V277T | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_K109N_T254V_V277T | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E | |||
| homo sapiens | OR1A2 | Q9Y585 | A108G_K109N_V205I_T254V_V277T | MKKENQSFNLDFILL ... | (R)-(-)-Carvone | 439570 | ULDHMXUKGWMISQ-SECBINFHSA-N | CC1=CC[C@H](CC1=O)C(=C)C | mono | 0 | norm_pair | 2000 | uM | 3 | Luc | HEK | liquid | in vitro | olf | rtp1s gγ13 | glosensor-22f | rho | C. Geithe, J. Protze, F. Kreuc ... | https://doi.org/10.1007/s00018 ... | Fig_S3E |